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Found 14 of ic50 data for polymerid = 50003824
TargetPyruvate kinase(Leishmania mexicana)
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50597707(CHEMBL5171047)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of Leishmania mexicana PYK (Asn75, Il61, Ser362, Arg73, Gln329 residues) incubated for 15 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPyruvate kinase(Leishmania mexicana)
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50270352((2S,3S,4S,5R)-N-cycloheptyl-5-((cycloheptylamino)m...)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of Leishmania mexicana pyruvate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase(Leishmania mexicana)
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50270448((2S,3S,4S,5R)-5-((cycloheptylamino)methyl)-3,4-dih...)
Affinity DataIC50:  5.30E+4nMAssay Description:Inhibition of Leishmania mexicana pyruvate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase(Leishmania mexicana)
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50270344(2,5-Anhydro-1-deoxy-1-(cycloheptylamino)-D-mannito...)
Affinity DataIC50:  7.10E+4nMAssay Description:Inhibition of Leishmania mexicana pyruvate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase(Leishmania mexicana)
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50270341((2R,3S,4S,5R)-2-(hydroxymethyl)-5-(((R)-1-(4-metho...)
Affinity DataIC50:  9.00E+5nMAssay Description:Inhibition of Leishmania mexicana pyruvate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase(Leishmania mexicana)
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50270338((2R,3S,4S,5R)-2-(hydroxymethyl)-5-((1,2,3,4-tetrah...)
Affinity DataIC50:  1.20E+6nMAssay Description:Inhibition of Leishmania mexicana pyruvate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase(Leishmania mexicana)
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50270349((2R,3S,4S,5R)-2-(hydroxymethyl)-5-(((R)-1-(naphtha...)
Affinity DataIC50:  1.50E+6nMAssay Description:Inhibition of Leishmania mexicana pyruvate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase(Leishmania mexicana)
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50270347((2R,3S,4S,5R)-2-(((1R,2S,4R)-bicyclo[2.2.1]heptan-...)
Affinity DataIC50:  1.50E+6nMAssay Description:Inhibition of Leishmania mexicana pyruvate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase(Leishmania mexicana)
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50270343((2R,3S,4S,5R)-2-(hydroxymethyl)-5-(((S)-1-(naphtha...)
Affinity DataIC50:  1.50E+6nMAssay Description:Inhibition of Leishmania mexicana pyruvate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase(Leishmania mexicana)
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50270345((2R,3S,4S,5R)-2-(hydroxymethyl)-5-(((S)-3-methylbu...)
Affinity DataIC50:  2.30E+6nMAssay Description:Inhibition of Leishmania mexicana pyruvate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase(Leishmania mexicana)
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50270474((2R,3S,4S,5R)-2-(hydroxymethyl)-5-((pentan-2-ylami...)
Affinity DataIC50:  2.50E+6nMAssay Description:Inhibition of Leishmania mexicana pyruvate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase(Leishmania mexicana)
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50270340((2R,3S,4S,5R)-2-(hydroxymethyl)-5-(((S)-1-(4-metho...)
Affinity DataIC50:  3.50E+6nMAssay Description:Inhibition of Leishmania mexicana pyruvate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase(Leishmania mexicana)
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50270449((2R,3S,4S,5R)-2-((cyclopentylamino)methyl)-5-(hydr...)
Affinity DataIC50:  4.10E+6nMAssay Description:Inhibition of Leishmania mexicana pyruvate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase(Leishmania mexicana)
Central University Of Punjab

Curated by ChEMBL
LigandPNGBDBM50270339((2R,3S,4S,5R)-2-((cyclobutylamino)methyl)-5-(hydro...)
Affinity DataIC50:  4.30E+6nMAssay Description:Inhibition of Leishmania mexicana pyruvate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed